SCHEMBL571306

SCHEMBL571306

CC(C)(C)OC(=O)NC1C[C@H](C(=O)O)C[C@@H]1O[Si](C)(C)C(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.48
KDM1A O60341 2/20 0.36
GAA P10253 1/20 0.35
MAOB P27338 2/20 0.35
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
KMT2A Q03164 2/20 0.33
MAOA P21397 1/20 0.33
CYP2C9 P11712 1/20 0.32
HSD11B1 P28845 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CTSK P43235 2/20 0.32
HDAC4 P56524 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1369991 1.00 BTK (0.48) BTKKDM1AGAAMAOBNFKB1
SCHEMBL31601158 1.00 BTK (0.48) BTKKDM1AGAAMAOBNFKB1
SCHEMBL30473209 0.91 BTK (0.51) BTKKDM1AGAAMAOBNFKB1
SCHEMBL31601203 0.87 BTK (0.37) BTKKDM1AGAAMAOBNFKB1
SCHEMBL15777845 0.82 BTK (0.61) BTKKDM1AGAAMAOBNFKB1
SCHEMBL31601393 0.82 KDM1A (0.40) BTKKDM1AGAAMAOBNFKB1
SCHEMBL31601395 0.82 KDM1A (0.40) BTKKDM1AGAAMAOBNFKB1
SCHEMBL4479750 0.82 BTK (0.39) BTKKDM1AGAAMAOBNFKB1
SCHEMBL30473133 0.82 BTK (0.39) BTKKDM1AGAAMAOBNFKB1
SCHEMBL4479752 0.82 BTK (0.39) BTKKDM1AGAAMAOBNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011044498-A9 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-02-09 WO disclosed
WO-2011044498-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2011-04-14 WO disclosed
WO-2010132839-A2 AMINOGLYCOSIDE DOSING REGIMENS ACHAOGEN, INC. (US) 2010-11-18 WO disclosed