SCHEMBL5720231

SCHEMBL5720231

CCC(C)C(C(=O)NC(Cc1ccccc1)C(O)CN(Cc1ccc(-c2ccccn2)cc1)NC(=O)C(NC(=O)O)C(C)(C)C)N1CCN(Cc2ccnnc2)C1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UGT1A1 P22309 3/20 0.58
MLNR O43193 1/20 0.58
NR1I2 O75469 1/20 0.58
SLCO2B1 O94956 1/20 0.58
ABCB11 O95342 1/20 0.58
ABCB1 P08183 1/20 0.58
CCKAR P32238 1/20 0.58
OPRK1 P41145 1/20 0.58
GHSR Q92847 1/20 0.58
SLCO1B3 Q9NPD5 1/20 0.58
ABCG2 Q9UNQ0 1/20 0.58
SLCO1B1 Q9Y6L6 1/20 0.58
CTSD P07339 4/20 0.52
CYP3A4 P08684 3/20 0.52
KCNH2 Q12809 1/20 0.46
CTSE P14091 1/20 0.33
PGC P20142 1/20 0.33
BRS3 P32247 1/20 0.31
CA2 P00918 1/20 0.31
BACE1 P56817 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3546338 1.00 UGT1A1 (0.58) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL9983143 1.00 UGT1A1 (0.58) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL3548730 0.95 UGT1A1 (0.66) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL3547902 0.94 UGT1A1 (0.59) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL3550738 0.94 UGT1A1 (0.58) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL3552706 0.92 UGT1A1 (0.60) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL5720601 0.92 UGT1A1 (0.60) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL3549386 0.91 UGT1A1 (0.58) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL3546919 0.90 UGT1A1 (0.57) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL3555056 0.90 UGT1A1 (0.67) UGT1A1MLNRNR1I2SLCO2B1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697348-A1 HIV PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 2006-09-06 EP claimed
WO-2005061487-A1 HIV PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 2005-07-07 WO claimed
EP-1697348-A1 HIV PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 2006-09-06 EP disclosed
WO-2005061487-A1 HIV PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 2005-07-07 WO disclosed