SCHEMBL5722017

SCHEMBL5722017

O=C(Cc1nccn1CC(=O)c1cccc(F)c1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.49
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA3 P07451 2/20 0.49
CA4 P22748 2/20 0.49
CA6 P23280 2/20 0.49
CA5A P35218 2/20 0.49
CA7 P43166 2/20 0.49
CA9 Q16790 2/20 0.49
CA13 Q8N1Q1 2/20 0.49
CA14 Q9ULX7 2/20 0.49
CA5B Q9Y2D0 2/20 0.49
ALPG P10696 5/20 0.46
PLAA Q9Y263 3/20 0.46
ALPL P05186 3/20 0.45
MGAM O43451 2/20 0.42
AMY1A P0DUB6 2/20 0.42
GAA P10253 2/20 0.42
SI P14410 2/20 0.42
MGAM2 Q2M2H8 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5722000 0.89 ALPG (0.45) CA12CA1CA2CA3CA4
SCHEMBL5721975 0.89 CA12 (0.51) CA12CA1CA2CA3CA4
SCHEMBL5721969 0.89 CA12 (0.53) CA12CA1CA2CA3CA4
SCHEMBL5721949 0.85 CA12 (0.54) CA12CA1CA2CA3CA4
SCHEMBL5721917 0.81 ALPG (0.46) CA12CA1CA2CA3CA4
SCHEMBL5722026 0.79 CA12 (0.73) CA12CA1CA2CA3CA4
SCHEMBL5721986 0.78 ALPG (0.47) CA12CA1CA2CA3CA4
SCHEMBL5722027 0.77 ALPG (0.49) CA12CA1CA2CA3CA4
SCHEMBL5722116 0.77 CA12 (0.55) CA12CA1CA2CA3CA4
SCHEMBL5722028 0.76 ALPG (0.50) CA12CA1CA2CA3CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554253-A4 IMIDAZOLIUM CXCR3 INHIBITORS SMITHKLINE BEECHAM CORP (US) 2006-09-20 EP disclosed
EP-1554253-A1 IMIDAZOLIUM CXCR3 INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2005-07-20 EP disclosed
WO-2003101970-A1 IMIDAZOLIUM CXCR3 INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-12-11 WO disclosed