SCHEMBL5725955

SCHEMBL5725955

OCC/C(=C(\c1ccc(O)cc1)c1ccc(Cl)cc1)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 13/20 0.61
ESRRG P62508 10/20 0.56
CYP19A1 P11511 4/20 0.56
ESR2 Q92731 3/20 0.56
ESRRB O95718 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5726578 1.00 ESR1 (0.61) ESR1ESRRGCYP19A1ESR2ESRRB
SCHEMBL5725960 1.00 ESR1 (0.61) ESR1ESRRGCYP19A1ESR2ESRRB
SCHEMBL1151880 0.92 ESR1 (0.71) ESR1ESRRGCYP19A1ESR2ESRRB
SCHEMBL1151987 0.92 ESR1 (0.71) ESR1ESRRGCYP19A1ESR2ESRRB
SCHEMBL1151986 0.92 ESR1 (0.71) ESR1ESRRGCYP19A1ESR2ESRRB
SCHEMBL5725055 0.92 ESR1 (0.71) ESR1ESRRGCYP19A1ESR2ESRRB
SCHEMBL2229348 0.92 ESR1 (0.71) ESR1ESRRGCYP19A1ESR2ESRRB
SCHEMBL1151879 0.92 ESR1 (0.71) ESR1ESRRGCYP19A1ESR2ESRRB
SCHEMBL5736018 0.87 ESR1 (0.63) ESR1ESRRGCYP19A1ESR2ESRRB
SCHEMBL5737374 0.87 ESR1 (0.63) ESR1ESRRGCYP19A1ESR2ESRRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1705169-A2 Triphenylalkene derivatives and their use as selective estrogen receptor modulators Hormos Medical Ltd. (FI) 2006-09-27 EP disclosed
EP-1235776-B1 TRIPHENYLALKENE DERIVATIVES AND THEIR USE AS SELECTIVE ESTROGEN RECEPTOR MODULATORS HORMOS MEDICAL CORP (FI) 2006-02-08 EP disclosed
US-6875775-B2 Triphenylalkene derivatives and their use as selective estrogen receptor modulators HORMOS MEDICAL OY LTD (FI) 2005-04-05 US disclosed
US-20030225130-A1 Triphenylalkene derivatives and their use as selective estrogen receptor modulators HORMOS MEDICAL OY LTD. 2003-12-04 US disclosed
US-6576645-B1 Such as 3-(4-chloro-1-(4-(2-(2-hydroxyethoxy)ethoxy)phenyl)--2-phenylbut-1 -enyl)phenol; producing tissue specific estro-genic and/or antiestrogenic effect HORMOS MEDICAL OY LTD (FI) 2003-06-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030225130-A1 Triphenylalkene derivatives and their use as selective estrogen receptor modulators ESR2, ESR1, GPER1 ESR1 2/4885ESRRG 6/4885CYP19A1 11/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.