SCHEMBL5727014

SCHEMBL5727014

Nc1nc(Nc2ccc(S(N)(=O)=O)cc2)nn1C(=O)c1cccnc1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 8/20 0.80
CDK1 P06493 8/20 0.80
CCNB1 P14635 8/20 0.80
CCNB3 Q8WWL7 8/20 0.80
JAK2 O60674 10/20 0.72
CCNA2 P20248 4/20 0.67
CDK2 P24941 4/20 0.67
CDK4 P11802 3/20 0.67
CCND1 P24385 3/20 0.67
MAPK3 P27361 3/20 0.67
MAPK1 P28482 3/20 0.67
KDR P35968 3/20 0.67
CSNK1A1 P48729 3/20 0.67
CSNK1D P48730 3/20 0.67
CSNK1E P49674 3/20 0.67
GSK3A P49840 3/20 0.67
GSK3B P49841 3/20 0.67
CSNK1G2 P78368 3/20 0.67
CCNA1 P78396 3/20 0.67
CSNK1G1 Q9HCP0 3/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5726202 0.89 CCNB2 (1.00) CCNB2CDK1CCNB1CCNB3JAK2
SCHEMBL5726369 0.88 CCNB2 (0.81) CCNB2CDK1CCNB1CCNB3JAK2
SCHEMBL1248065 0.86 JAK1 (0.64) CCNB2CDK1CCNB1CCNB3JAK2
SCHEMBL24339597 0.84 JAK2 (1.00) CCNB2CDK1CCNB1CCNB3JAK2
SCHEMBL6099748 0.83 CCNB2 (0.81) CCNB2CDK1CCNB1CCNB3JAK2
SCHEMBL6102584 0.83 CCNB2 (0.77) CCNB2CDK1CCNB1CCNB3JAK2
SCHEMBL6102916 0.83 CCNB2 (0.87) CCNB2CDK1CCNB1CCNB3JAK2
SCHEMBL5986060 0.82 CCNB2 (0.79) CCNB2CDK1CCNB1CCNB3JAK2
SCHEMBL4037292 0.81 CCNB2 (0.70) CCNB2CDK1CCNB1CCNB3JAK2
SCHEMBL6101578 0.81 CCNB2 (0.74) CCNB2CDK1CCNB1CCNB3JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1712550-A2 Substituted triazole diamine derivatives as kinase inhibitors Ortho-McNeil Pharmaceutical, Inc. (US) 2006-10-18 EP disclosed
EP-1355889-B1 SUBSTITUTED TRIAZOLE DIAMINE DERIVATIVES AS KINASE INHIBITORS ORTHO MCNEIL PHARM INC (US) 2006-06-07 EP disclosed