SCHEMBL5736044

SCHEMBL5736044

CN(C)CCOc1cccc(-c2ccnc(NCc3ccc(C(=O)Nc4ccccc4N)cc3)n2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 17/20 1.00
HDAC3 O15379 4/20 0.65
HDAC2 Q92769 4/20 0.65
NCOR1 O75376 3/20 0.65
CYP3A4 P08684 1/20 0.65
HDAC11 Q96DB2 1/20 0.65
HDAC8 Q9BY41 1/20 0.65
HDAC6 Q9UBN7 1/20 0.65
NCOR2 Q9Y618 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL211036 0.99 HDAC1 (0.98) HDAC1HDAC3HDAC2NCOR1CYP3A4
SCHEMBL209388 0.91 HDAC1 (1.00) HDAC1HDAC3HDAC2NCOR1CYP3A4
SCHEMBL13593882 0.90 HDAC1 (0.82) HDAC1HDAC3HDAC2NCOR1CYP3A4
SCHEMBL212798 0.88 HDAC1 (0.79) HDAC1HDAC3HDAC2NCOR1CYP3A4
SCHEMBL209215 0.85 HDAC1 (0.73) HDAC1HDAC3HDAC2NCOR1CYP3A4
SCHEMBL211058 0.84 HDAC1 (0.75) HDAC1HDAC3HDAC2NCOR1CYP3A4
SCHEMBL212310 0.83 HDAC1 (1.00) HDAC1HDAC3HDAC2NCOR1CYP3A4
SCHEMBL2732829 0.83 HDAC1 (0.85) HDAC1HDAC3HDAC2NCOR1CYP3A4
SCHEMBL212106 0.81 HDAC1 (0.80) HDAC1HDAC3HDAC2NCOR1CYP3A4
SCHEMBL1064494 0.80 HDAC1 (1.00) HDAC1HDAC3HDAC2NCOR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1735319-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2006-12-27 EP disclosed
WO-2005092899-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2005-10-06 WO disclosed