SCHEMBL5736233

SCHEMBL5736233

Nc1ccccc1NC(=O)c1ccc(CNc2nc3ccc(OCCC4CCCCN4)cc3s2)cc1

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 11/20 0.68
AURKB Q96GD4 7/20 0.67
HDAC3 O15379 2/20 0.47
HDAC2 Q92769 1/20 0.47
SCD O00767 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL211854 0.85 HDAC1 (0.78) HDAC1AURKBHDAC3HDAC2SCD
SCHEMBL213867 0.83 HDAC1 (0.86) HDAC1AURKB
SCHEMBL210479 0.81 HDAC1 (0.77) HDAC1AURKBSCD
SCHEMBL209760 0.81 HDAC1 (0.85) HDAC1AURKB
SCHEMBL1061039 0.81 HDAC1 (1.00) HDAC1AURKB
SCHEMBL1064488 0.80 HDAC1 (1.00) HDAC1SCD
SCHEMBL13390247 0.79 HDAC1 (0.79) HDAC1AURKB
SCHEMBL214421 0.77 HDAC1 (0.82) HDAC1HDAC3HDAC2
SCHEMBL210213 0.76 HDAC1 (0.81) HDAC1HDAC3HDAC2SCD
SCHEMBL2733826 0.76 HDAC1 (0.79) HDAC1HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1735319-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2006-12-27 EP disclosed
WO-2005092899-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2005-10-06 WO disclosed