SCHEMBL573945

SCHEMBL573945

Cn1cc(-c2cc(Oc3ccc(F)c(NC(=O)Nc4cc(N5CCCC5)cc(C(F)(F)F)c4)c3)ccn2)cn1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 17/20 0.56
BRAF P15056 4/20 0.49
CSF1R P07333 4/20 0.47
MET P08581 3/20 0.47
PDGFRB P09619 3/20 0.47
PDGFRA P16234 3/20 0.47
FLT3 P36888 2/20 0.47
NTRK1 P04629 1/20 0.45
KIT P10721 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL574104 0.99 KDR (0.55) KDRBRAFCSF1RMETPDGFRB
SCHEMBL573458 0.95 KDR (0.55) KDRBRAFCSF1RMETPDGFRB
SCHEMBL573559 0.94 KDR (0.56) KDRBRAFCSF1RMETPDGFRB
SCHEMBL859861 0.94 KDR (0.54) KDRBRAFCSF1RMETPDGFRB
SCHEMBL574063 0.93 KDR (0.55) KDRBRAFCSF1RMETPDGFRB
SCHEMBL573467 0.91 KDR (0.56) KDRCSF1RMETPDGFRBPDGFRA
SCHEMBL573433 0.91 KDR (0.52) KDRBRAFCSF1RMETPDGFRB
SCHEMBL826931 0.91 KDR (0.48) KDRBRAFCSF1RMETPDGFRB
SCHEMBL573312 0.90 KDR (0.56) KDRCSF1RMETPDGFRBPDGFRA
SCHEMBL574300 0.90 KDR (0.52) KDRCSF1RMETPDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012019015-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF MYELOPROLIFERATIVE DISEASES AND OTHER PROLIFERATIVE DISEASES DECIPHERA PHARMACEUTICALS, LLC (US) 2012-02-09 WO disclosed
US-20110189167-A1 Methods and Compositions for the Treatment of Myeloproliferative Diseases and other Proliferative Diseases DECIPHERA PHARMACEUTICALS, LLC 2011-08-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110189167-A1 Methods and Compositions for the Treatment of Myeloproliferative Diseases and other Proliferative Diseases MCL1, NRAS, ABL1 KDR 2434/4885BRAF 12/4885CSF1R 1244/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.