SCHEMBL5739587

SCHEMBL5739587

CNc1cc(Oc2ccc3c(C(=O)Nc4c[nH]c(=O)c(C)c4)cccc3c2)ccn1

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.70
FGFR1 P11362 12/20 0.53
CSF1R P07333 1/20 0.49
FGFR2 P21802 1/20 0.49
FGFR3 P22607 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4548897 0.85 KDR (0.84) KDRFGFR1CSF1RFGFR2FGFR3
SCHEMBL4548900 0.84 KDR (0.76) KDRFGFR1FGFR2FGFR3
SCHEMBL4548908 0.83 KDR (0.71) KDRFGFR1FGFR2FGFR3
SCHEMBL2748198 0.83 KDR (0.84) KDRFGFR1CSF1RFGFR2
SCHEMBL4548898 0.82 KDR (1.00) KDRFGFR1CSF1RFGFR2FGFR3
SCHEMBL4548899 0.81 KDR (0.75) KDRFGFR1
SCHEMBL4548910 0.81 KDR (0.84) KDRFGFR1CSF1RFGFR2FGFR3
SCHEMBL22540525 0.81 KDR (0.74) KDRFGFR1CSF1RFGFR2FGFR3
SCHEMBL2747256 0.81 KDR (0.74) KDRFGFR1CSF1RFGFR2FGFR3
SCHEMBL4548901 0.81 KDR (0.79) KDRFGFR1CSF1RFGFR2FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1713484-A2 COMPOUNDS AND METHODS OF USE AMGEN INC. (US) 2006-10-25 EP disclosed
WO-2005070891-A2 COMPOUNDS AND METHODS OF USE AMGEN INC (US) 2005-08-04 WO disclosed