SCHEMBL5739893

SCHEMBL5739893

COC(=O)Oc1cn2ncnc(Nc3cccc(O)c3)c2c1C

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDR P35968 15/20 0.71
EGFR P00533 3/20 0.49
ERBB2 P04626 1/20 0.46
RET P07949 1/20 0.44
FGFR1 P11362 1/20 0.44
FLT1 P17948 1/20 0.44
CDK2 P24941 1/20 0.44
PIK3R1 P27986 1/20 0.44
EPHB2 P29323 1/20 0.44
KIF5B P33176 1/20 0.44
TTBK1 Q5TCY1 1/20 0.44
NOD1 Q9Y239 1/20 0.43
MAP2K1 Q02750 1/20 0.43
MAPK14 Q16539 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5739937 0.88 KDR (0.56) KDREGFRERBB2MAPK14
SCHEMBL5739216 0.87 KDR (0.55) KDREGFRERBB2MAP2K1MAPK14
SCHEMBL5739989 0.87 KDR (0.53) KDREGFRRETKIF5BMAP2K1
SCHEMBL5740244 0.86 KDR (0.54) KDREGFRERBB2RETMAP2K1
SCHEMBL5739549 0.86 KDR (0.54) KDREGFRERBB2MAPK14
SCHEMBL5740324 0.86 KDR (0.54) KDREGFRERBB2MAP2K1MAPK14
SCHEMBL5739951 0.86 KDR (0.71) KDREGFRFLT1
SCHEMBL5739127 0.85 KDR (0.56) KDRMAPK14
SCHEMBL5740240 0.85 KDR (0.53) KDREGFRERBB2MAPK14
SCHEMBL5740103 0.85 KDR (0.59) KDREGFRMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed