SCHEMBL574061

SCHEMBL574061

NC(=O)Nc1ccc(Oc2ccnc(-c3cnn(CCO)c3)c2)cc1F

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AXL P30530 1/20 0.48
CSF1R P07333 13/20 0.45
PDGFRA P16234 7/20 0.45
PDGFRB P09619 6/20 0.45
MET P08581 5/20 0.45
KDR P35968 5/20 0.45
FLT3 P36888 4/20 0.45
KIT P10721 3/20 0.41
FEN1 P39748 1/20 0.41
FGFR1 P11362 1/20 0.41
NAMPT P43490 1/20 0.41
IKBKE Q14164 1/20 0.40
TBK1 Q9UHD2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2898454 0.93 AXL (0.51) AXLCSF1RPDGFRAPDGFRBMET
SCHEMBL2919897 0.87 AXL (0.60) AXLCSF1RPDGFRAPDGFRBMET
SCHEMBL574161 0.82 KDR (0.49) AXLCSF1RPDGFRAPDGFRBMET
SCHEMBL574737 0.82 KDR (0.60) AXLCSF1RPDGFRAPDGFRBMET
SCHEMBL827559 0.82 MAPK14 (0.47) AXLCSF1RPDGFRAPDGFRBMET
SCHEMBL827920 0.82 MAPK14 (0.65) AXLCSF1RPDGFRAMETKDR
SCHEMBL574452 0.81 KDR (0.54) AXLCSF1RPDGFRAPDGFRBMET
SCHEMBL574521 0.81 AXL (0.46) AXLCSF1RPDGFRAPDGFRBMET
SCHEMBL574062 0.81 MAPK14 (0.63) AXLKDR
SCHEMBL3665924 0.79 AXL (0.61) AXLCSF1RPDGFRAPDGFRBMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012019015-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF MYELOPROLIFERATIVE DISEASES AND OTHER PROLIFERATIVE DISEASES DECIPHERA PHARMACEUTICALS, LLC (US) 2012-02-09 WO disclosed