SCHEMBL5741282

SCHEMBL5741282

CCOC(=O)OC(=O)C(=CN(C)C)C(=O)c1ccccc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
KDM4E B2RXH2 2/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
CYP11B2 P19099 3/20 0.38
TSHR P16473 2/20 0.38
MAPT P10636 4/20 0.37
CYP1A2 P05177 3/20 0.37
CYP2C19 P33261 3/20 0.37
CYP2C9 P11712 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
LMNA P02545 2/20 0.37
ALDH1A1 P00352 3/20 0.36
CYP3A4 P08684 1/20 0.36
GAA P10253 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2953731 0.91 CYP11B1 (0.50) CYP11B1SMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL29398562 0.91 CYP11B1 (0.50) CYP11B1SMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL2953727 0.91 CYP11B1 (0.50) CYP11B1SMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL6016300 0.91 CYP11B1 (0.50) CYP11B1SMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL3446933 0.85 CYP11B1 (0.47) CYP11B1SMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL29058653 0.80 CYP11B1 (0.52) CYP11B1SMN1; SMN2NPC1KDM4ECES2
SCHEMBL15962343 0.79 CYP11B1 (0.51) CYP11B1SMN1; SMN2NPC1CES2CES1
SCHEMBL2282849 0.78 MEN1 (0.44) CYP11B1SMN1; SMN2KDM4ECES2CES1
SCHEMBL1931607 0.78 MEN1 (0.44) CYP11B1SMN1; SMN2KDM4ECES2CES1
SCHEMBL3570354 0.78 KMT2A (0.50) CYP11B1SMN1; SMN2NPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1727820-A2 AMINE DERIVATIVES MERCK PATENT GmbH (DE) 2006-12-06 EP disclosed
WO-2005054246-A2 AMINE DERIVATIVES HAVING A TYROSINE-KINASE-INHIBITING EFFECT MERCK PATENT GMBH (DE) 2005-06-16 WO disclosed