SCHEMBL5741963

SCHEMBL5741963

COc1ccc(S(=O)(=O)N2CCN(CCc3nc(N4CC(C)CC(C)C4)c4ccccc4n3)CC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 10/20 0.56
HSD11B1 P28845 1/20 0.50
LMNA P02545 1/20 0.50
PKM P14618 4/20 0.45
ALDH1A1 P00352 2/20 0.45
KMT2A Q03164 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
NPC1 O15118 1/20 0.43
USP2 O75604 1/20 0.43
CFTR P13569 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5741797 0.91 GBA1 (0.54) GBA1HSD11B1LMNAPKMALDH1A1
SCHEMBL5789177 0.91 GBA1 (0.59) GBA1HSD11B1LMNAPKMALDH1A1
SCHEMBL5743384 0.89 GBA1 (0.63) GBA1HSD11B1LMNAPKMALDH1A1
SCHEMBL5740458 0.89 GBA1 (0.60) GBA1HSD11B1LMNAPKMALDH1A1
SCHEMBL5742174 0.88 GBA1 (0.62) GBA1HSD11B1LMNAPKMALDH1A1
SCHEMBL5741175 0.87 GBA1 (0.64) GBA1HSD11B1LMNAPKMALDH1A1
SCHEMBL5741406 0.86 GBA1 (0.58) GBA1HSD11B1LMNAPKMALDH1A1
SCHEMBL5742978 0.86 GBA1 (0.54) GBA1HSD11B1LMNAPKMALDH1A1
SCHEMBL5743497 0.86 GBA1 (0.57) GBA1HSD11B1LMNAPKMALDH1A1
SCHEMBL5740505 0.85 GBA1 (0.56) GBA1HSD11B1LMNAPKMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1646615-A1 PYRIMIDINE DERIVATIVES AS MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2006-04-19 EP disclosed
WO-2004111014-A1 PYRIMIDINE DERIVATIVES AS MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2004-12-23 WO disclosed