SCHEMBL5744809

SCHEMBL5744809

COc1ccc2ncc(Cl)c([C@H](O)CN3CCC(N)CC3)c2n1

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.50
SLC2A1 P11166 4/20 0.41
PTPN11 Q06124 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5744804 1.00 KCNH2 (0.50) KCNH2SLC2A1PTPN11
SCHEMBL5744806 1.00 KCNH2 (0.50) KCNH2SLC2A1PTPN11
SCHEMBL5746247 0.88 KCNH2 (0.42) KCNH2PTPN11
SCHEMBL5440972 0.84 PTPN11 (0.45) KCNH2PTPN11
SCHEMBL5744343 0.81 KCNH2 (0.49) KCNH2SLC2A1
SCHEMBL5252383 0.81 KCNH2 (0.60) KCNH2SLC2A1
SCHEMBL5256971 0.81 KCNH2 (0.60) KCNH2SLC2A1
SCHEMBL5256973 0.81 KCNH2 (0.60) KCNH2SLC2A1
Hydrochloric Acid SCHEMBL5253585 0.80 KCNH2 (0.59) KCNH2SLC2A1
SCHEMBL5744136 0.78 KCNH2 (0.61) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1578743-A4 ANTIBACTERIAL AGENTS GLAXO GROUP LTD (GB) 2006-11-29 EP disclosed
EP-1578743-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2005-09-28 EP disclosed
WO-2004058144-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2004-07-15 WO disclosed