SCHEMBL574499

SCHEMBL574499

COc1cc(N2CCC(N(S(C)(=O)=O)S(C)(=O)=O)C(C)(C)C2)ccc1Nc1ncc(Cl)c(-c2c[nH]c3ccccc23)n1

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 2/20 0.69
EGFR P00533 14/20 0.66
IGF1R P08069 5/20 0.50
KCNH2 Q12809 3/20 0.47
INSR P06213 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL518359 0.91 ALK (0.74) ALKEGFRIGF1RKCNH2
SCHEMBL517766 0.88 ALK (0.75) ALKEGFRIGF1RKCNH2
SCHEMBL517604 0.87 ALK (0.81) ALKEGFRIGF1RKCNH2
SCHEMBL518394 0.82 ALK (0.83) ALKEGFRIGF1RKCNH2INSR
SCHEMBL29355191 0.82 ALK (1.00) ALKEGFRIGF1RKCNH2
SCHEMBL517412 0.82 ALK (1.00) ALKEGFRIGF1RKCNH2
SCHEMBL518078 0.82 EGFR (0.83) ALKEGFRIGF1RINSR
SCHEMBL517293 0.82 ALK (0.84) ALKEGFRIGF1RKCNH2
SCHEMBL518047 0.82 ALK (0.84) ALKEGFRIGF1RKCNH2
SCHEMBL10207758 0.82 ALK (0.59) ALKEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2601186-A2 4-(1H-INDOL-3-YL)-PYRIMIDINES AS ALK INHIBITORS AstraZeneca AB (SE) 2013-06-12 EP disclosed
WO-2012017239-A2 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2012-02-09 WO disclosed