SCHEMBL5748880

SCHEMBL5748880

CCCCNS(=O)(=O)c1cccc(Nc2ncnn3cc(OC(=O)OC)c(C)c23)c1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.47
EGFR P00533 1/20 0.42
ERBB2 P04626 1/20 0.42
MAPK14 Q16539 7/20 0.42
TNNI3K Q59H18 1/20 0.40
PIK3CD O00329 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CG P48736 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045967 0.87 KDR (0.65) KDREGFRERBB2MAPK14
SCHEMBL5740324 0.85 KDR (0.54) KDREGFRERBB2MAPK14
SCHEMBL5740240 0.85 KDR (0.53) KDREGFRERBB2MAPK14TNNI3K
SCHEMBL5740244 0.80 KDR (0.54) KDREGFRERBB2MAPK14
SCHEMBL5739216 0.79 KDR (0.55) KDREGFRERBB2MAPK14
SCHEMBL5739937 0.78 KDR (0.56) KDREGFRERBB2MAPK14
SCHEMBL5739127 0.78 KDR (0.56) KDRMAPK14
SCHEMBL5741956 0.77 KDR (0.67) KDREGFRMAPK14
SCHEMBL5739549 0.77 KDR (0.54) KDREGFRERBB2MAPK14
SCHEMBL5740103 0.76 KDR (0.59) KDREGFRMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed