SCHEMBL5752565

SCHEMBL5752565

CNCCCn1nc(C2=C(c3cn(C)c4ccc(Cl)cc34)C(=O)NC2=O)c2ccccc21

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 14/20 0.54
GSK3A P49840 2/20 0.54
MEN1 O00255 1/20 0.54
RGS12 O14924 1/20 0.54
GMNN O75496 1/20 0.54
USP2 O75604 1/20 0.54
CCNB2 O95067 1/20 0.54
LMNA P02545 1/20 0.54
TP53 P04637 1/20 0.54
CYP1A2 P05177 1/20 0.54
CDK1 P06493 1/20 0.54
POLB P06746 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
MAPT P10636 1/20 0.54
CYP2C9 P11712 1/20 0.54
CDK4 P11802 1/20 0.54
CCNB1 P14635 1/20 0.54
NFKB1 P19838 1/20 0.54
CCNA2 P20248 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3775916 0.90 GSK3B (0.58) GSK3BGSK3AMEN1RGS12GMNN
SCHEMBL3781580 0.89 GSK3B (0.66) GSK3BGSK3AMEN1RGS12GMNN
SCHEMBL5757844 0.88 GSK3B (0.67) GSK3BGSK3AMEN1RGS12GMNN
SCHEMBL5754334 0.86 GSK3B (0.67) GSK3BGSK3AMEN1RGS12GMNN
SCHEMBL5754325 0.85 GSK3B (0.69) GSK3BGSK3AMEN1RGS12GMNN
SCHEMBL3771143 0.85 GSK3B (0.52) GSK3BGSK3AMEN1RGS12GMNN
SCHEMBL1128498 0.85 GSK3B (0.52) GSK3BGSK3AMEN1RGS12GMNN
SCHEMBL1127704 0.84 IDH1 (0.70) GSK3BIDH1
SCHEMBL4689265 0.84 GSK3B (0.50) GSK3BGSK3AMEN1RGS12GMNN
SCHEMBL4691089 0.84 GSK3B (0.50) GSK3BGSK3AMEN1RGS12GMNN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362047-B1 INDAZOLYL-SUBSTITUTED PYRROLINE COMPOUNDS AS KINASE INHIBITORS ORTHO MCNEIL PHARM INC (US) 2006-05-17 EP disclosed