SCHEMBL5754277

SCHEMBL5754277

COc1ccc(-c2cc(CC(=O)OC(C)C)n[nH]2)cc1C1CCCO1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 3/20 0.34
FLT3 P36888 1/20 0.34
NTRK3 Q16288 1/20 0.34
NTRK2 Q16620 1/20 0.34
OXTR P30559 3/20 0.33
AVPR1A P37288 3/20 0.33
NPC1 O15118 1/20 0.33
CASP3 P42574 1/20 0.33
RAB9A P51151 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
PDE4B Q07343 1/20 0.32
MAPK8 P45983 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3606197 0.76 BRD4 (0.36) OXTRAVPR1ANPC1CASP3RAB9A
SCHEMBL5755289 0.74 ADORA2A (0.37)
SCHEMBL5756897 0.64 PDE4B (0.41) NPC1RAB9AALDH1A1KDM4EHSD17B10
SCHEMBL4197982 0.61 PDE4B (0.48) PDE4B
SCHEMBL3010672 0.60 ABL1 (0.58) NPC1KMT2AALDH1A1CYP1A2CYP3A4
SCHEMBL14532521 0.60 NPY5R (0.51) NPY5RALDH1A1KDM4ECYP1A2HSD17B10
SCHEMBL30949067 0.60 HTR2C (0.47) KMT2ATDP1
SCHEMBL13304474 0.59 KDM4E (0.37) NPC1RAB9AALDH1A1KDM4ECYP1A2
SCHEMBL5184733 0.58 PDE4B (0.42) NPY5RALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL21767410 0.58 CFTR (0.45) OXTRAVPR1AKMT2AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1631568-A1 PYRAZOLE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS Memory Pharmaceuticals Corporation (US) 2006-03-08 EP claimed
WO-2004094411-A1 PYRAZOLE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS MEMORY PHARMACEUTICALS CORPORATION (US) 2004-11-04 WO claimed
EP-1631568-A1 PYRAZOLE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS Memory Pharmaceuticals Corporation (US) 2006-03-08 EP disclosed
WO-2004094411-A1 PYRAZOLE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS MEMORY PHARMACEUTICALS CORPORATION (US) 2004-11-04 WO disclosed