SCHEMBL5758328

SCHEMBL5758328

CS(=O)(=O)OCCCc1cccc(OCc2coc(/C=C/c3ccccc3)n2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 8/20 0.40
MGLL Q99685 1/20 0.39
CYSLTR2 Q9NS75 3/20 0.39
CYSLTR1 Q9Y271 3/20 0.39
LCK P06239 1/20 0.39
ERBB2 P04626 1/20 0.39
MINK1 Q8N4C8 1/20 0.39
PPARG P37231 4/20 0.37
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
CCNB2 O95067 1/20 0.35
CDK1 P06493 1/20 0.35
CDK4 P11802 1/20 0.35
CCNB1 P14635 1/20 0.35
CCND1 P24385 1/20 0.35
CCNB3 Q8WWL7 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
PKM P14618 1/20 0.35
CYP4F2 P78329 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5758332 1.00 PPARA (0.40) PPARAMGLLCYSLTR2CYSLTR1LCK
SCHEMBL5762449 0.90 ERBB2 (0.47) PPARAMGLLCYSLTR2CYSLTR1ERBB2
SCHEMBL5762454 0.90 ERBB2 (0.47) PPARAMGLLCYSLTR2CYSLTR1ERBB2
SCHEMBL5762604 0.88 ERBB2 (0.49) PPARAMGLLCYSLTR2CYSLTR1ERBB2
SCHEMBL5757663 0.88 ERBB2 (0.49) PPARAMGLLCYSLTR2CYSLTR1ERBB2
SCHEMBL5761048 0.87 ERBB2 (0.49) PPARAMGLLCYSLTR2CYSLTR1ERBB2
SCHEMBL5757306 0.87 ERBB2 (0.49) PPARAMGLLCYSLTR2CYSLTR1ERBB2
SCHEMBL5761043 0.87 ERBB2 (0.49) PPARAMGLLCYSLTR2CYSLTR1ERBB2
SCHEMBL5757310 0.87 ERBB2 (0.49) PPARAMGLLCYSLTR2CYSLTR1ERBB2
SCHEMBL5756640 0.85 MAPT (0.38) ERBB2MINK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1270571-B1 Heterocyclic compounds, their production and use TAKEDA PHARMACEUTICAL (JP) 2006-09-06 EP disclosed
EP-1270571-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-01-02 EP disclosed
US-6211215-B1 AROMATIC HETEROCYCLIC COMPOUND WITH AZOLE COMPOUND TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed
EP-0912562-A1 HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1999-05-06 EP disclosed
WO-1998003505-A2 HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-01-29 WO disclosed