SCHEMBL5759422

SCHEMBL5759422

C(=Cc1nc(COc2ccc(CCCCn3ccnn3)cc2)co1)c1ccccc1

nearest known ligand 0.80

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 2/20 0.80
MINK1 Q8N4C8 1/20 0.80
ATP4A P20648 9/20 0.40
ATP4B P51164 9/20 0.40
FFAR1 O14842 3/20 0.39
CYSLTR2 Q9NS75 1/20 0.35
CYSLTR1 Q9Y271 1/20 0.35
HMOX1 P09601 1/20 0.34
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33
LCK P06239 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5759417 1.00 ERBB2 (0.80) ERBB2MINK1ATP4AATP4BFFAR1
SCHEMBL5759321 0.97 ERBB2 (0.75) ERBB2MINK1ATP4AATP4BFFAR1
SCHEMBL5759315 0.97 ERBB2 (0.75) ERBB2MINK1ATP4AATP4BFFAR1
SCHEMBL28473428 0.93 ERBB2 (0.82) ERBB2MINK1ATP4AATP4BFFAR1
SCHEMBL22398131 0.93 ERBB2 (0.82) ERBB2MINK1ATP4AATP4BFFAR1
SCHEMBL27688109 0.93 ERBB2 (0.82) ERBB2MINK1ATP4AATP4BFFAR1
SCHEMBL28480663 0.92 ERBB2 (0.81) ERBB2MINK1ATP4AATP4BFFAR1
SCHEMBL22397926 0.92 ERBB2 (0.81) ERBB2MINK1ATP4AATP4BFFAR1
SCHEMBL22398145 0.91 ERBB2 (0.72) ERBB2MINK1ATP4AATP4BFFAR1
SCHEMBL28472667 0.91 ERBB2 (0.72) ERBB2MINK1ATP4AATP4BFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1270571-B1 Heterocyclic compounds, their production and use TAKEDA PHARMACEUTICAL (JP) 2006-09-06 EP disclosed
EP-1270571-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-01-02 EP disclosed
US-6211215-B1 AROMATIC HETEROCYCLIC COMPOUND WITH AZOLE COMPOUND TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed