SCHEMBL5760447

SCHEMBL5760447

COCCCN[C@H]1CCN(C(=O)O)C1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
EPHX2 P34913 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
CYP3A4 P08684 1/20 0.40
KDM4E B2RXH2 3/20 0.39
MCHR1 Q99705 2/20 0.38
CHRM2 P08172 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM3 P20309 1/20 0.38
GAA P10253 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
LMNA P02545 2/20 0.37
SMYD3 Q9H7B4 1/20 0.37
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4503490 0.91 KDM4E (0.40) TSHRSMN1; SMN2KDM4EMCHR1CHRM2
SCHEMBL4877080 0.81 KDM4E (0.45) TSHRSMN1; SMN2KDM4ECHRM2CHRM5
SCHEMBL25208208 0.81 PARP1 (0.43) EPHX2SMN1; SMN2KDM4EMCHR1CHRM2
SCHEMBL23152417 0.81 PARP1 (0.43) EPHX2SMN1; SMN2KDM4EMCHR1CHRM2
SCHEMBL4117382 0.81 PARP1 (0.43) EPHX2SMN1; SMN2KDM4EMCHR1CHRM2
SCHEMBL31580602 0.80 DPP7 (0.37) KDM4EMCHR1SMYD3
SCHEMBL3833559 0.76 EPHX2 (0.39) EPHX2CYP3A4KDM4ECHRM2CHRM5
SCHEMBL3827038 0.76 EPHX2 (0.39) EPHX2CYP3A4KDM4ECHRM2CHRM5
SCHEMBL18115895 0.76 EPHX2 (0.39) EPHX2CYP3A4KDM4ECHRM2CHRM5
SCHEMBL5996911 0.75 TSHR (0.55) TSHREPHX2SMN1; SMN2CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638934-A1 3-AMINOPYRROLIDINES AS INHIBITORS OF MONOAMINE UPTAKE ELI LILLY AND COMPANY (US) 2006-03-29 EP disclosed
WO-2005000811-A1 3-AMINOPYRROLIDINES AS INHIBITORS OF MONOAMINE UPTAKE ELI LILLY AND COMPANY (US) 2005-01-06 WO disclosed