SCHEMBL5761971

SCHEMBL5761971

Cc1ccccc1-c1cc(N2CCC(OCCO)CC2)ncc1OC(=O)N(C)Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 17/20 0.57
CYP3A4 P08684 2/20 0.48
GPBAR1 Q8TDU6 1/20 0.46
SGMS1 Q86VZ5 1/20 0.40
SGMS2 Q8NHU3 1/20 0.40
SMO Q99835 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5763724 0.90 TACR1 (0.61) TACR1CYP3A4GPBAR1
SCHEMBL7086321 0.88 TACR1 (0.74) TACR1CYP3A4GPBAR1SGMS1SGMS2
SCHEMBL5761333 0.81 TACR1 (0.56) TACR1CYP3A4
SCHEMBL3880526 0.77 TACR1 (0.61) TACR1GPBAR1
SCHEMBL6525284 0.76 TACR1 (0.81) TACR1CYP3A4GPBAR1
SCHEMBL905366 0.76 TACR1 (0.73) TACR1CYP3A4GPBAR1SGMS1SGMS2
SCHEMBL5779738 0.75 TACR1 (0.59) TACR1GPBAR1
SCHEMBL905394 0.75 TACR1 (0.79) TACR1CYP3A4GPBAR1
SCHEMBL5760285 0.75 SMO (0.46) TACR1CYP3A4SMO
SCHEMBL905343 0.74 TACR1 (0.78) TACR1CYP3A4GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1305319-B1 4-PHENYL-PYRIDINE DERIVATIVES AS NEUROKININ-1 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2006-04-05 EP claimed