SCHEMBL5762046

SCHEMBL5762046

Cc1ccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 14/20 1.00
FGFR1 P11362 11/20 1.00
PDGFRB P09619 10/20 1.00
PDGFRA P16234 10/20 1.00
ABL1 P00519 8/20 1.00
MAPK14 Q16539 8/20 1.00
EGFR P00533 8/20 1.00
WEE1 P30291 3/20 0.84
FGFR2 P21802 1/20 0.84
FGFR4 P22455 1/20 0.84
FGFR3 P22607 1/20 0.84
KIT P10721 3/20 0.83
PSEN1 P49768 1/20 0.80
PSEN2 P49810 1/20 0.80
APH1B Q8WW43 1/20 0.80
NCSTN Q92542 1/20 0.80
APH1A Q96BI3 1/20 0.80
PSENEN Q9NZ42 1/20 0.80
ACVR1 Q04771 2/20 0.78
RIPK2 O43353 1/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17520126 0.95 SRC (0.90) SRCFGFR1PDGFRBPDGFRAABL1
SCHEMBL5764062 0.93 FGFR1 (1.00) SRCFGFR1PDGFRBPDGFRAABL1
SCHEMBL1249524 0.91 FGFR1 (1.00) SRCFGFR1PDGFRBPDGFRAABL1
SCHEMBL11939526 0.91 FGFR1 (0.84) SRCFGFR1PDGFRBPDGFRAABL1
SCHEMBL13498143 0.91 FGFR1 (0.83) SRCFGFR1PDGFRBPDGFRAABL1
SCHEMBL1334768 0.91 SRC (1.00) SRCFGFR1PDGFRBPDGFRAABL1
SCHEMBL2083696 0.91 SRC (1.00) SRCFGFR1PDGFRBPDGFRAABL1
SCHEMBL2081574 0.91 SRC (1.00) SRCFGFR1PDGFRBPDGFRAABL1
SCHEMBL868353 0.89 FGFR1 (1.00) SRCFGFR1PDGFRBPDGFRAABL1
SCHEMBL4747103 0.89 SRC (0.81) SRCFGFR1PDGFRBPDGFRAABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0823908-B1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2006-11-02 EP claimed
WO-2005105097-A2 PYRIDOPYRIMIDINES FOR TREATING INFLAMMATORY AND OTHER DISEASES GPC BIOTECH AG (DE) 2005-11-10 WO claimed
EP-0823908-A1 PYRIDO 2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1998-02-18 EP claimed
WO-1996034867-A1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1996-11-07 WO claimed
EP-0823908-B1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2006-11-02 EP disclosed
WO-2005105097-A2 PYRIDOPYRIMIDINES FOR TREATING INFLAMMATORY AND OTHER DISEASES GPC BIOTECH AG (DE) 2005-11-10 WO disclosed