SCHEMBL5764908

SCHEMBL5764908

Cn1c(=O)c(-c2c(Cl)cccc2Cl)cc2cnc(NCc3ccccc3)nc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 14/20 1.00
ABL1 P00519 7/20 0.81
EGFR P00533 7/20 0.78
SRC P12931 5/20 0.74
FGFR2 P21802 2/20 0.74
FGFR4 P22455 2/20 0.74
FGFR3 P22607 2/20 0.74
WEE1 P30291 1/20 0.74
PDGFRB P09619 2/20 0.69
PDGFRA P16234 2/20 0.69
MAPK14 Q16539 2/20 0.69
KIT P10721 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5762106 0.90 FGFR1 (1.00) FGFR1ABL1EGFRSRCFGFR2
SCHEMBL5764474 0.88 FGFR1 (1.00) FGFR1ABL1EGFRSRCFGFR2
SCHEMBL2248398 0.87 FGFR1 (0.76) FGFR1ABL1EGFRSRCFGFR2
SCHEMBL5763078 0.87 FGFR1 (1.00) FGFR1ABL1EGFRSRCFGFR2
SCHEMBL5762061 0.85 FGFR1 (1.00) FGFR1ABL1EGFRSRCFGFR2
SCHEMBL1249524 0.85 FGFR1 (1.00) FGFR1ABL1EGFRSRCFGFR2
SCHEMBL5762058 0.84 FGFR1 (1.00) FGFR1ABL1EGFRSRCFGFR2
SCHEMBL5763919 0.84 FGFR1 (1.00) FGFR1ABL1EGFRSRCFGFR2
SCHEMBL14014657 0.82 FGFR1 (0.70) FGFR1ABL1EGFRSRCFGFR2
SCHEMBL5763583 0.82 FGFR1 (1.00) FGFR1ABL1EGFRSRCFGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0823908-B1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2006-11-02 EP claimed
WO-2005105097-A2 PYRIDOPYRIMIDINES FOR TREATING INFLAMMATORY AND OTHER DISEASES GPC BIOTECH AG (DE) 2005-11-10 WO claimed
EP-0823908-A1 PYRIDO 2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1998-02-18 EP claimed
WO-1996034867-A1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1996-11-07 WO claimed
EP-0823908-B1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2006-11-02 EP disclosed
WO-2005105097-A2 PYRIDOPYRIMIDINES FOR TREATING INFLAMMATORY AND OTHER DISEASES GPC BIOTECH AG (DE) 2005-11-10 WO disclosed