SCHEMBL5766271

SCHEMBL5766271

CCn1c(=O)c(-c2cc(Cl)ccc2Cl)cc2cnc(NCCCN3CCN(C)CC3)nc21

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 10/20 0.62
SRC P12931 4/20 0.62
EGFR P00533 3/20 0.62
FGFR2 P21802 2/20 0.62
FGFR4 P22455 2/20 0.62
FGFR3 P22607 2/20 0.62
PAK1 Q13153 5/20 0.60
PKN1 Q16512 4/20 0.60
PAK4 O96013 3/20 0.60
SIK2 Q9H0K1 3/20 0.56
SIK1 P57059 1/20 0.56
SIK3 Q9Y2K2 1/20 0.56
WEE1 P30291 1/20 0.53
PAK2 Q13177 4/20 0.51
MAPK8 P45983 1/20 0.49
STK26 Q9P289 2/20 0.48
STK24 Q9Y6E0 2/20 0.48
STK4 Q13043 1/20 0.48
STK3 Q13188 1/20 0.48
PAK3 O75914 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5764398 0.87 FGFR1 (0.82) FGFR1SRCEGFRFGFR2FGFR4
SCHEMBL5762258 0.77 FGFR1 (1.00) FGFR1SRCEGFRFGFR2FGFR4
SCHEMBL15580670 0.76 PAK1 (0.64) FGFR1EGFRPAK1PKN1PAK4
SCHEMBL5764642 0.74 FGFR1 (1.00) FGFR1SRCEGFRFGFR2FGFR4
SCHEMBL16195710 0.74 PKN1 (0.62) FGFR1SRCEGFRFGFR2FGFR4
SCHEMBL5763017 0.74 FGFR1 (1.00) FGFR1SRCEGFRFGFR2FGFR4
SCHEMBL15036161 0.72 PAK1 (0.73) FGFR1SRCEGFRFGFR2FGFR4
SCHEMBL15281586 0.72 PAK1 (0.72) FGFR1SRCEGFRFGFR2FGFR4
SCHEMBL29593396 0.71 MAPK8 (0.74) FGFR1SRCEGFRFGFR2FGFR4
SCHEMBL14014812 0.71 MAPK8 (0.75) FGFR1SRCEGFRFGFR2FGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0823908-B1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2006-11-02 EP claimed