SCHEMBL5773454

SCHEMBL5773454

CCOC(=O)Cc1c(C#N)ccc(N(CC(F)(F)C2=NC(C)=CCC2=O)C(=O)C(F)(F)F)c1F

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.33
CYP2C9 P11712 1/20 0.33
AR P10275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3886853 0.78 F2 (0.44) KDM4ECYP2C9
SCHEMBL5773458 0.77 F2 (0.38) KDM4ECYP2C9
SCHEMBL3890749 0.76 F2 (0.32) KDM4ECYP2C9
SCHEMBL13792116 0.75 F2 (0.44)
SCHEMBL5771914 0.70 F2 (0.43)
SCHEMBL3888694 0.69 KDM4E (0.45) KDM4ECYP2C9
SCHEMBL5774527 0.64 F2 (0.53)
SCHEMBL31682816 0.63 KDM4E (0.40) KDM4EAR
SCHEMBL4332770 0.61 RXFP1 (0.39) KDM4EAR
SCHEMBL3888182 0.60 F2 (0.66) KDM4ECYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613319-A2 SUBSTITUTED PHENYL ACETAMIDES AND THEIR USE AS PROTEASE INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-01-11 EP disclosed
WO-2004091613-A2 SUBSTITUTED PHENYL ACETAMIDES AND THEIR USE AS PROTEASE INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2004-10-28 WO disclosed