SCHEMBL5774174

SCHEMBL5774174

O=c1nc(-c2ccncc2)oc2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.48
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
ATAD2 Q6PL18 1/20 0.46
ELANE P08246 1/20 0.45
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
PIK3CB P42338 2/20 0.44
PIK3CA P42336 1/20 0.44
HSD17B10 Q99714 3/20 0.43
TSHR P16473 1/20 0.43
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 2/20 0.42
MAPT P10636 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TP53 P04637 1/20 0.42
PKM P14618 1/20 0.42
GLA P06280 1/20 0.42
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL812662 0.89 NPC1 (0.53) NPC1RAB9AELANEHSD17B10ALDH1A1
SCHEMBL4029088 0.87 ELANE (0.58) NPC1RAB9AELANEHSD17B10TSHR
SCHEMBL30025603 0.87 ELANE (0.58) NPC1RAB9AELANEHSD17B10TSHR
SCHEMBL4028915 0.84 ELANE (0.54) NPC1RAB9AELANEHSD17B10TSHR
SCHEMBL7869611 0.84 NPC1 (0.51) NPC1RAB9AELANEHSD17B10ALDH1A1
SCHEMBL2882726 0.83 NPC1 (0.58) NPC1RAB9AHSD17B10ALDH1A1KDM4E
SCHEMBL5307439 0.81 NPC1 (0.60) NPC1RAB9AELANEHSD17B10TSHR
SCHEMBL311688 0.81 NPC1 (0.54) NPC1RAB9AHSD17B10ALDH1A1KDM4E
SCHEMBL3791447 0.81 NPC1 (0.63) NPC1RAB9AELANEHSD17B10ALDH1A1
SCHEMBL5307520 0.81 TNKS (0.54) NPC1RAB9AELANEALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558260-A4 QUINAZOLINONE COMPOUNDS AS CALCILYTICS NPS PHARMA INC (US) 2006-10-25 EP disclosed
EP-1558260-A2 QUINAZOLINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2005-08-03 EP disclosed
WO-2004041755-A2 QUINAZOLINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2004-05-21 WO disclosed