SCHEMBL5778550

SCHEMBL5778550

Cc1ccnc(NCC2CCNCC2)n1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 4/20 0.59
PAK4 O96013 1/20 0.54
PAK1 Q13153 1/20 0.54
BRD4 O60885 3/20 0.51
ATAD2 Q6PL18 2/20 0.51
AXL P30530 1/20 0.44
FLT3 P36888 1/20 0.44
TYRO3 Q06418 1/20 0.44
MERTK Q12866 1/20 0.44
GAS6 Q14393 1/20 0.44
ROCK2 O75116 2/20 0.42
TRIM58 Q8NG06 2/20 0.42
ROCK1 Q13464 1/20 0.42
CDC42BPB Q9Y5S2 1/20 0.42
VCP P55072 1/20 0.41
CDC7 O00311 2/20 0.41
CDK2 P24941 2/20 0.41
CCNB2 O95067 1/20 0.41
MAP4K4 O95819 1/20 0.41
CDK1 P06493 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13402933 0.89 HRH4 (0.55) HRH4PAK4PAK1ROCK2VCP
SCHEMBL13403220 0.85 CDC7 (0.51) HRH4PAK4PAK1ROCK2VCP
SCHEMBL13493639 0.84 HRH4 (0.50) HRH4PAK4PAK1ROCK2VCP
SCHEMBL761678 0.79 HRH4 (0.54) HRH4PAK4PAK1BRD4ATAD2
Hydrochloric Acid SCHEMBL6152965 0.78 HRH4 (0.54) HRH4PAK4PAK1BRD4ATAD2
SCHEMBL1914496 0.78 HRH4 (0.51) HRH4PAK4PAK1BRD4ATAD2
SCHEMBL6508763 0.77 IKBKB (0.58) HRH4BRD4ATAD2FLT3CDK2
SCHEMBL27886899 0.77 HRH4 (0.50) HRH4PAK4PAK1BRD4ATAD2
SCHEMBL27886901 0.76 HRH4 (0.52) HRH4PAK4PAK1BRD4ATAD2
Hydrochloric Acid SCHEMBL6582848 0.75 BRD4 (0.50) HRH4PAK4PAK1BRD4ATAD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379520-B1 N-SUBSTITUTED NONARYL-HETEROCYCLIC NMDA/NR2B ANTAGONISTS MERCK & CO INC (US) 2006-04-26 EP disclosed