SCHEMBL5778607

SCHEMBL5778607

Cn1cncc1C(c1ccc(Cl)cc1)c1ccc2nc(OC(=O)NC3CC3)cc(-c3cccc(Cl)c3)c2c1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FNTA P49354 9/20 0.56
FNTB P49356 9/20 0.56
PGGT1B P53609 8/20 0.38
PTGS2 P35354 1/20 0.36
NPR1 P16066 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5783326 0.87 FNTA (0.58) FNTAFNTBPGGT1BNPR1
SCHEMBL5781151 0.85 FNTA (0.54) FNTAFNTBPGGT1B
SCHEMBL5780208 0.85 FNTA (0.52) FNTAFNTBPGGT1B
SCHEMBL5782193 0.85 FNTA (0.54) FNTAFNTBPGGT1B
SCHEMBL5782042 0.85 FNTA (0.54) FNTAFNTBPGGT1B
SCHEMBL5784774 0.83 FNTA (0.51) FNTAFNTBPGGT1B
SCHEMBL5782628 0.83 FNTA (0.52) FNTAFNTBPGGT1B
SCHEMBL5779856 0.82 FNTA (0.54) FNTAFNTBPGGT1B
SCHEMBL5783128 0.81 FNTA (0.66) FNTAFNTBPGGT1B
Hydrochloric Acid SCHEMBL5780158 0.79 FNTA (0.64) FNTAFNTBPGGT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322635-B1 FARNESYL TRANSFERASE INHIBITING QUINOLINE AND QUINAZOLINE DERIVATIVES AS FARNESYL TRANSFERASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2006-03-22 EP claimed