SCHEMBL5779074

SCHEMBL5779074

CN1CCN(Cc2cccc(CN3Cc4c(NC(=O)C5=CC(Cl)=CCC5=S)cccc4C3=O)c2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 3/20 0.45
BTK Q06187 1/20 0.38
SUCNR1 Q9BXA5 2/20 0.36
HDAC1 Q13547 3/20 0.36
CDK5 Q00535 1/20 0.35
DYRK1A Q13627 1/20 0.35
CDK5R1 Q15078 1/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
DHPS P49366 1/20 0.35
ACHE P22303 1/20 0.34
KIT P10721 1/20 0.34
KDR P35968 1/20 0.34
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5781280 0.92 F10 (0.46) F10HDAC1CDK5DYRK1ACDK5R1
SCHEMBL5782217 0.89 F10 (0.46) F10HDAC1DHPSALDH1A1HDAC3
SCHEMBL5777471 0.89 F10 (0.48) F10HDAC1DHPSALDH1A1MEN1
SCHEMBL5782626 0.88 F10 (0.50) F10HDAC1PDCD1CD274DHPS
SCHEMBL5783180 0.88 F10 (0.48) F10HDAC1DHPSALDH1A1HDAC3
SCHEMBL5779859 0.88 F10 (0.48) F10HDAC1DHPSALDH1A1MEN1
SCHEMBL5784062 0.87 F10 (0.47) F10HDAC1DHPSALDH1A1MEN1
SCHEMBL5783769 0.86 F10 (0.48) F10HDAC1PDCD1CD274DHPS
SCHEMBL5784722 0.85 F10 (0.49) F10HDAC1DHPSALDH1A1HDAC3
SCHEMBL5783655 0.85 F10 (0.45) F10HDAC1DHPSALDH1A1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1408962-B1 SUBSTITUTED ISOINDOLES AND THE USE THEREOF BAYER HEALTHCARE AG (DE) 2006-03-15 EP disclosed
EP-1408962-A1 SUBSTITUTED ISOINDOLES AND THE USE THEREOF Bayer HealthCare AG (DE) 2004-04-21 EP disclosed
WO-2003007942-A1 SUBSTITUTED ISOINDOLES AND THE USE THEREOF BAYER HEALTHCARE AG (DE) 2003-01-30 WO disclosed