SCHEMBL5779310

SCHEMBL5779310

Cc1cc2ccc(-c3cccc4ccccc34)cc2cc1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.46
ACMSD Q8TDX5 1/20 0.46
ENPP3 O14638 1/20 0.46
ENPP1 P22413 1/20 0.46
TLR8 Q9NR97 1/20 0.46
ALDH1A1 P00352 2/20 0.45
CYP2A6 P11509 2/20 0.45
CA12 O43570 4/20 0.44
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CA9 Q16790 4/20 0.44
CYP1A2 P05177 3/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25177116 0.89 MCL1 (0.51) MCL1ACMSDENPP3ENPP1ALDH1A1
SCHEMBL29195637 0.89 MCL1 (0.51) MCL1ACMSDENPP3ENPP1ALDH1A1
SCHEMBL1470544 0.89 MCL1 (0.51) MCL1ACMSDENPP3ENPP1ALDH1A1
SCHEMBL29986101 0.89 MCL1 (0.51) MCL1ACMSDENPP3ENPP1ALDH1A1
SCHEMBL31742566 0.89 MCL1 (0.54) MCL1ACMSDENPP3ENPP1ALDH1A1
SCHEMBL598962 0.87 GSTP1 (0.57) MCL1ACMSDENPP3ENPP1ALDH1A1
SCHEMBL30274189 0.87 GSTP1 (0.57) MCL1ACMSDENPP3ENPP1ALDH1A1
SCHEMBL3176171 0.82 GSTP1 (0.61) MCL1ACMSDALDH1A1CYP1A2HPGD
SCHEMBL12344996 0.82 CYP2A6 (0.50) MCL1ACMSDTLR8ALDH1A1CYP2A6
SCHEMBL1527419 0.81 HPRT1 (0.54) MCL1ACMSDALDH1A1CYP2A6CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615890-A1 PIPERIDINE DERIVATIVES AS RENIN INHIBITORS FOR THE TREATMENT OF HYPERTENSION WARNER-LAMBERT COMPANY (US) 2006-01-18 EP disclosed
WO-2004089903-A1 PIPERIDINE DERIVATIVES AS RENIN INHIBITORS FOR THE TREATMENT OF HYPERTENSION WARNER-LAMBERT COMPANY LLC (US) 2004-10-21 WO disclosed