SCHEMBL5785482

SCHEMBL5785482

Nc1nc(NC(Cc2ccc(Cl)cc2)C2CCCN2)nc2nc(-c3ccco3)nn12

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.55
ADORA1 P30542 7/20 0.55
ADORA3 P0DMS8 6/20 0.55
ADORA2B P29275 3/20 0.52
ALDH1A1 P00352 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
MAPK1 P28482 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
TMEM97 Q5BJF2 1/20 0.49
HSD17B10 Q99714 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5785842 0.89 ADORA2A (0.54) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL5787999 0.85 ADORA2A (0.57) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL5784479 0.82 ADORA2A (0.49) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL9327254 0.76 ADORA2A (0.81) ADORA2AADORA1ADORA3ADORA2BALDH1A1
SCHEMBL6010026 0.76 ADORA2A (0.45) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL5410869 0.75 ADORA2A (0.62) ADORA2AADORA1ADORA3ADORA2BALDH1A1
SCHEMBL6010465 0.74 ADORA2A (0.37) ADORA2AADORA1
SCHEMBL6009997 0.73 ADORA2A (0.44) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL5418880 0.73
SCHEMBL6009814 0.73 ADORA2A (0.38) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615930-A2 TRIAZOLOTRIAZINES AND PYRAZOLOTRIAZINES USEFUL AS A2A ADENOSINE RECEPTOR ANTAGONISTS Biogen Idec MA, Inc. (US) 2006-01-18 EP claimed
WO-2004092170-A2 TRIAZOLOTRIAZINES AND PYRAZOLOTRIAZINES USEFUL AS A2A ADENOSINE RECEPTOR ANTAGON ISTS BIOGEN IDEC MA INC. (US) 2004-10-28 WO claimed