SCHEMBL5790840

SCHEMBL5790840

Cc1ccc(C(=O)O)c(-n2ccnn2)c1-n1ccnn1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.41
HCRTR1 O43613 6/20 0.41
HCRTR2 O43614 6/20 0.41
HAAO P46952 1/20 0.37
CMA1 P23946 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL302594 0.86 HCRTR1 (0.40) NOTUMHCRTR1HCRTR2ALDH1A1
SCHEMBL1586907 0.86 HCRTR1 (0.53) NOTUMHCRTR1HCRTR2CMA1ALDH1A1
SCHEMBL29160361 0.80 NOTUM (0.45) NOTUMHCRTR1HCRTR2ALDH1A1
SCHEMBL9286585 0.80 NOTUM (0.40) NOTUMHCRTR1HCRTR2CMA1
SCHEMBL18016687 0.77 NOTUM (0.51) NOTUMCMA1ALDH1A1
SCHEMBL27883266 0.75 HCRTR1 (0.54) NOTUMHCRTR1HCRTR2ALDH1A1
SCHEMBL17028392 0.75 NOTUM (0.41) NOTUMHCRTR1HCRTR2ALDH1A1
SCHEMBL1670997 0.75 HCRTR1 (0.53) HCRTR1HCRTR2ALDH1A1
SCHEMBL1586336 0.74 HCRTR1 (0.55) HCRTR1HCRTR2
SCHEMBL5790843 0.74 NOTUM (0.47) NOTUMHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1725544-A1 3-[4-HETEROCYCLYL-1,2,3-TRIAZOL-1-YL]-N-ARYL-BENZAMIDES AS INHIBITORS OF THE CYTOKINES PRODUCTION FOR THE TREATMENT OF CHRONIC INFLAMMATORY DISEASES BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2006-11-29 EP disclosed
WO-2005090333-A1 3-‘4-HETEROCYCLYL -1,2,3,-TRIAZOL-1-YL!-N-ARYL-BENZAMIDES AS INHIBITORS OF THE CYTOKINES PRODUCTION FOR THE TREATMENT OF CHRONIC INFLAMMATORY DISEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-09-29 WO disclosed