SCHEMBL5792216

SCHEMBL5792216

COc1ccc(F)cc1C(C)(O)CC(N)OCc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 8/20 0.43
NR3C1 P04150 17/20 0.42
TACR1 P25103 1/20 0.41
PGR P06401 2/20 0.39
CETP P11597 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5791756 0.89 TACR1 (0.41) NR3C1TACR1CETP
SCHEMBL5793713 0.89 TACR1 (0.47) NR3C2NR3C1TACR1CETP
SCHEMBL5790053 0.87 TACR1 (0.42) NR3C2NR3C1TACR1CETP
SCHEMBL5791612 0.85 TACR1 (0.42) TACR1CETP
SCHEMBL5821974 0.84 TACR1 (0.44) TACR1CETP
SCHEMBL5793395 0.83 TACR1 (0.49) TACR1CETP
SCHEMBL5792826 0.83 TACR1 (0.41) TACR1CETP
SCHEMBL5790666 0.81 TACR1 (0.47) TACR1CETP
SCHEMBL5793711 0.79 TACR1 (0.47) TACR1CETP
SCHEMBL5793709 0.79 TACR1 (0.47) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006014942-A1 ARYLOXYALKYLAMINE NK-1/SSRI INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-02-09 WO claimed
WO-2006014942-A1 ARYLOXYALKYLAMINE NK-1/SSRI INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-02-09 WO disclosed