SCHEMBL5797574

SCHEMBL5797574

Nc1nc(N)c2c(n1)c(I)c(-c1cccc(CCC(=O)O)c1)c1[nH]ccc12

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 11/20 0.43
CDK2 P24941 1/20 0.37
PPARG P37231 1/20 0.37
IKBKB O14920 1/20 0.35
CHUK O15111 1/20 0.35
DHFR P00374 5/20 0.35
PLA2G10 O15496 1/20 0.35
PLA2G2A P14555 1/20 0.35
SLCO1B1 Q9Y6L6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5796955 0.88 FFAR1 (0.36) FFAR1PPARGDHFR
SCHEMBL5795879 0.82 PARP1 (0.38) DHFR
SCHEMBL4690844 0.81 PLA2G10 (0.40) FFAR1CDK2PPARGDHFRPLA2G10
SCHEMBL5799326 0.81 FFAR1 (0.43) FFAR1DHFRPLA2G10
SCHEMBL4691250 0.71 MAP4K4 (0.42) FFAR1IKBKBCHUKDHFR
SCHEMBL4691075 0.71 CDK2 (0.48) CDK2IKBKBCHUKDHFRPLA2G10
SCHEMBL5798206 0.69
SCHEMBL4693946 0.67 PARP1 (0.42) DHFR
SCHEMBL4688624 0.64 FFAR1 (0.40) FFAR1DHFRPLA2G10PLA2G2ASLCO1B1
SCHEMBL21484487 0.64 FFAR1 (0.91) FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1628979-A1 DIAMINOPYRROLOQUINAZOLINES COMPOUNDS AS PROTEIN TYROSINE PHOSPHATASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2006-03-01 EP claimed
WO-2004101568-A1 DIAMINOPYRROLOQUINAZOLINES COMPOUNDS AS PROTEIN TYROSINE PHOSPHATASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2004-11-25 WO claimed