SCHEMBL5799335

SCHEMBL5799335

Cn1ncc(Br)c1Nc1ccc(-c2ccccc2)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.40
MEN1 O00255 2/20 0.40
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TTK P33981 3/20 0.38
DHODH Q02127 3/20 0.37
BRD4 O60885 1/20 0.36
BPTF Q12830 1/20 0.36
KAT2B Q92831 1/20 0.36
BRD9 Q9H8M2 1/20 0.36
HTR2A P28223 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5796502 0.91 MEN1 (0.43) KMT2AMEN1LMNASMN1; SMN2TTK
SCHEMBL4913037 0.79 KDM4E (0.50) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL4900772 0.79 KCNH2 (0.41) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL4901251 0.79 BCDIN3D (0.45) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL4910942 0.77 HTR2A (0.46) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL4913021 0.77 BRD4 (0.40) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL14281210 0.74 MEN1 (0.41) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL4909185 0.74 GAA (0.43) KMT2AMEN1MAPTSMN1; SMN2BRD4
SCHEMBL4909812 0.73 HTR2A (0.41) KMT2AMEN1HTR2A
SCHEMBL4908676 0.72 HTR2A (0.45) KMT2AMEN1KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006060762-A2 PYRAZOLE DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2006-06-08 WO disclosed