SCHEMBL5800599

SCHEMBL5800599

CN(CC(CCN1CC(N2CCC(O)CC2)C1)c1ccc(F)cc1)C(=O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 16/20 0.50
TACR1 P25103 1/20 0.44
KCNH2 Q12809 1/20 0.40
CCR5 P51681 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4257153 1.00 TACR2 (0.50) TACR2TACR1KCNH2CCR5
SCHEMBL4258295 0.94 TACR2 (0.51) TACR2TACR1KCNH2CCR5
SCHEMBL5798549 0.94 TACR2 (0.51) TACR2TACR1KCNH2CCR5
SCHEMBL4256226 0.91 TACR2 (0.49) TACR2TACR1KCNH2
SCHEMBL4256311 0.90 TACR2 (0.49) TACR2TACR1KCNH2CCR5
SCHEMBL4264167 0.89 TACR2 (0.65) TACR2
SCHEMBL5802168 0.89 TACR2 (0.65) TACR2
SCHEMBL4256282 0.88 TACR2 (0.47) TACR2TACR1KCNH2
SCHEMBL4255121 0.88 TACR2 (0.51) TACR2
SCHEMBL5799585 0.88 TACR2 (0.51) TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006062478-A1 NOVEL TREATMENT OF GASTROINTESTINAL DISORDERS ASTRAZENECA AB (SE) 2006-06-15 WO claimed