SCHEMBL5806983

SCHEMBL5806983

COc1ccc2ncc(F)c(CCN3CCC(NCc4ccc5c(n4)NC(=O)CO5)CC3)c2c1

nearest known ligand 0.77

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 16/20 0.77
KCNQ1 P51787 1/20 0.71
CACNA1C Q13936 1/20 0.71
SLC2A1 P11166 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6079771 0.99 KCNH2 (0.76) KCNH2KCNQ1CACNA1CSLC2A1
Hydrochloric Acid SCHEMBL5745009 0.91 KCNH2 (0.76) KCNH2KCNQ1CACNA1C
SCHEMBL6079668 0.90 KCNH2 (0.72) KCNH2KCNQ1CACNA1CSLC2A1
Hydrochloric Acid SCHEMBL5744101 0.90 KCNH2 (0.72) KCNH2KCNQ1CACNA1C
Hydrochloric Acid SCHEMBL5795282 0.90 KCNH2 (0.71) KCNH2KCNQ1CACNA1CSLC2A1
Hydrochloric Acid SCHEMBL6078820 0.89 KCNH2 (0.63) KCNH2KCNQ1CACNA1CSLC2A1
Hydrochloric Acid SCHEMBL6078814 0.89 KCNH2 (0.63) KCNH2KCNQ1CACNA1CSLC2A1
Hydrochloric Acid SCHEMBL6078808 0.89 KCNH2 (0.63) KCNH2KCNQ1CACNA1CSLC2A1
SCHEMBL3273196 0.88 KCNH2 (0.60) KCNH2KCNQ1CACNA1CSLC2A1
SCHEMBL13400404 0.86 KCNH2 (0.69) KCNH2KCNQ1CACNA1CSLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1578743-A4 ANTIBACTERIAL AGENTS GLAXO GROUP LTD (GB) 2006-11-29 EP disclosed
EP-1578743-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2005-09-28 EP disclosed
WO-2004058144-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2004-07-15 WO disclosed