SCHEMBL5807003

SCHEMBL5807003

Cn1c(=O)n(-c2ccccc2)c2nc(Nc3cccc(C(=O)O)c3)ncc21

nearest known ligand 0.76

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 5/20 0.76
PRKDC P78527 2/20 0.56
EGFR P00533 2/20 0.55
FGFR1 P11362 1/20 0.55
BTK Q06187 3/20 0.52
AURKA O14965 4/20 0.51
RHOA P61586 1/20 0.50
ADORA2A P29274 1/20 0.48
GSK3A P49840 1/20 0.48
PTK2 Q05397 1/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
CDK4 P11802 1/20 0.47
CCND1 P24385 1/20 0.47
CCND2 P30279 1/20 0.47
CCND3 P30281 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5803243 0.84 GSK3B (0.76) GSK3BPRKDCEGFRFGFR1BTK
SCHEMBL13763871 0.74 AURKA (0.78) GSK3BEGFRFGFR1AURKARHOA
SCHEMBL1599121 0.73 GSK3B (1.00) GSK3BPRKDCEGFRADORA2ACDK4
SCHEMBL5803855 0.73 GSK3B (1.00) GSK3BPRKDCEGFRFGFR1BTK
SCHEMBL5803009 0.73 GSK3B (0.72) GSK3BPRKDCEGFRFGFR1ADORA2A
SCHEMBL30030206 0.72 PRKDC (0.67) GSK3BPRKDCADORA2A
SCHEMBL30030843 0.72 PRKDC (0.67) GSK3BPRKDCADORA2A
SCHEMBL5815034 0.72 GSK3B (0.71) GSK3BPRKDCEGFRFGFR1BTK
SCHEMBL5764437 0.71 FGFR1 (1.00) EGFRFGFR1BTK
SCHEMBL29651071 0.70 GSK3B (0.64) GSK3BPRKDCADORA2AGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006091737-A1 MODULATORS OF GSK-3 ACTIVITY KEMIA, INC. (US) 2006-08-31 WO disclosed