SCHEMBL5807199

SCHEMBL5807199

CC(c1nc(N(C)C)c2ccccc2n1)N1CCN(S(=O)(=O)c2ccc(Br)cc2)CC1.CC(c1nc(N(C)C)c2ccccc2n1)N1CCN(S(=O)(=O)c2ccc(Br)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.53
GBA1 P04062 10/20 0.52
L3MBTL1 Q9Y468 1/20 0.43
MAPT P10636 1/20 0.43
USP2 O75604 2/20 0.41
LMNA P02545 2/20 0.41
MAPK1 P28482 2/20 0.41
HTT P42858 2/20 0.41
PKM P14618 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ADRA2A P08913 2/20 0.41
NPY5R Q15761 2/20 0.41
MCHR1 Q99705 2/20 0.41
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3823336 1.00 CFTR (0.53) CFTRGBA1L3MBTL1MAPTUSP2
SCHEMBL3819657 0.90 CFTR (0.53) CFTRGBA1L3MBTL1MAPTUSP2
SCHEMBL5820778 0.90 CFTR (0.53) CFTRGBA1L3MBTL1MAPTUSP2
SCHEMBL5804966 0.89 CFTR (0.51) CFTRGBA1L3MBTL1MAPTUSP2
SCHEMBL3823980 0.89 CFTR (0.51) CFTRGBA1L3MBTL1MAPTUSP2
SCHEMBL3818773 0.88 CFTR (0.68) CFTRGBA1LMNAHTTPKM
SCHEMBL13724387 0.84 CFTR (0.67) CFTRGBA1L3MBTL1MAPTUSP2
SCHEMBL3816463 0.84 CFTR (0.53) CFTRGBA1L3MBTL1MAPTUSP2
SCHEMBL3816459 0.83 CFTR (0.52) CFTRGBA1L3MBTL1MAPTUSP2
SCHEMBL3821009 0.83 CFTR (0.61) CFTRGBA1L3MBTL1MAPTUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1646615-A1 PYRIMIDINE DERIVATIVES AS MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2006-04-19 EP disclosed
WO-2004111014-A1 PYRIMIDINE DERIVATIVES AS MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2004-12-23 WO disclosed