Bicarbonate

Bicarbonate

SCHEMBL580920

COC(=O)c1ccnc(-c2ccc(C(F)(F)F)cc2C)c1.Cl.O=C([O-])[O-].[K+].[K+]

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.49
KDM4C Q9H3R0 3/20 0.49
KDM6B O15054 2/20 0.49
KDM5C P41229 2/20 0.49
KDM2A Q9Y2K7 2/20 0.49
KDM3A Q9Y4C1 2/20 0.49
TLR2 O60603 1/20 0.45
TLR1 Q15399 1/20 0.45
JMJD6 Q6NYC1 2/20 0.44
MRGPRX4 Q96LA9 1/20 0.44
KDM1A O60341 1/20 0.41
HDAC1 Q13547 1/20 0.41
PHGDH O43175 1/20 0.40
GPBAR1 Q8TDU6 1/20 0.40
LMNA P02545 1/20 0.40
CFTR P13569 1/20 0.40
KDM5B Q9UGL1 1/20 0.39
TRPV1 Q8NER1 2/20 0.39
MAOB P27338 1/20 0.39
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL580921 1.00 KDM4E (0.49) KDM4EKDM4CKDM6BKDM5CKDM2A
Hydrochloric Acid SCHEMBL580962 0.95 KDM4E (0.53) KDM4EKDM4CKDM6BKDM5CKDM2A
Hydrochloric Acid SCHEMBL581889 0.85 KDM4E (0.52) KDM4EKDM4CKDM6BKDM5CKDM2A
Hydrochloric Acid SCHEMBL581125 0.79 KDM4E (0.46) KDM4EKDM4CKDM6BKDM5CKDM2A
SCHEMBL581356 0.78 KDM4C (0.58) KDM4EKDM4CKDM6BKDM5CKDM2A
Hydrochloric Acid SCHEMBL582068 0.77 SYK (0.36) KDM4EKDM4CKDM6BKDM5CKDM2A
SCHEMBL14976243 0.76 KDM4C (0.51) KDM4EKDM4CKDM6BKDM5CKDM2A
SCHEMBL28490524 0.75 KDM4C (0.61) KDM4EKDM4CKDM6BKDM5CKDM2A
SCHEMBL581753 0.75 KDM4E (0.55) KDM4EKDM4CKDM6BKDM5CKDM2A
SCHEMBL30772297 0.75 KDM4E (0.55) KDM4EKDM4CKDM6BKDM5CKDM2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed