SCHEMBL5809213

SCHEMBL5809213

CC(C)c1c(C(=O)Nc2ccc(F)cc2)c(-c2ccccc2)c(-c2ccc(F)cc2)n1CCCN1CCOCC1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE6D O43924 3/20 0.68
HMGCR P04035 5/20 0.61
SLCO1B1 Q9Y6L6 4/20 0.61
ABCB11 O95342 3/20 0.61
HDAC1 Q13547 2/20 0.61
HDAC2 Q92769 2/20 0.61
HDAC6 Q9UBN7 2/20 0.61
NR1I2 O75469 1/20 0.61
RHOC P08134 1/20 0.61
CYP3A4 P08684 1/20 0.61
THRB P10828 1/20 0.61
NR1H4 Q96RI1 1/20 0.61
ABCG2 Q9UNQ0 1/20 0.61
ABCB1 P08183 1/20 0.60
ABCC2 Q92887 1/20 0.60
ABCC3 O15438 2/20 0.59
ABCC4 O15439 2/20 0.59
SLCO1B3 Q9NPD5 2/20 0.59
TRPV4 Q9HBA0 3/20 0.52
MAPK1 P28482 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14318916 0.99 PDE6D (0.69) PDE6DHMGCRSLCO1B1ABCB11HDAC1
SCHEMBL5809115 0.92 HMGCR (0.64) PDE6DHMGCRSLCO1B1ABCB11HDAC1
SCHEMBL5805276 0.91 HMGCR (0.65) PDE6DHMGCRSLCO1B1ABCB11HDAC1
SCHEMBL5804695 0.91 SLCO1B1 (0.64) PDE6DHMGCRSLCO1B1ABCB11HDAC1
SCHEMBL5809062 0.91 SLCO1B1 (0.64) PDE6DHMGCRSLCO1B1ABCB11HDAC1
SCHEMBL5804873 0.90 HMGCR (0.65) PDE6DHMGCRSLCO1B1ABCB11HDAC1
SCHEMBL5805228 0.88 HMGCR (0.67) PDE6DHMGCRSLCO1B1ABCB11HDAC1
SCHEMBL5804867 0.87 HMGCR (0.66) PDE6DHMGCRSLCO1B1ABCB11HDAC1
SCHEMBL5805022 0.87 SLCO1B1 (0.57) PDE6DHMGCRSLCO1B1ABCB11HDAC1
SCHEMBL4978670 0.86 PDE6D (0.78) PDE6DHMGCRSLCO1B1ABCB11HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006110918-A1 PYRROLE COMPOUNDS AND USES THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2006-10-19 WO claimed