SCHEMBL581127

SCHEMBL581127

COC(=O)C1CCNC(c2cc(F)c(C(F)(F)F)c(F)c2)C1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.35
SLC6A4 P31645 3/20 0.35
SLC6A3 Q01959 3/20 0.35
CHRNA1 P02708 1/20 0.35
CHRNG P07510 1/20 0.35
ITGA5 P08648 1/20 0.35
CHRNB1 P11230 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
CHRND Q07001 1/20 0.35
MAPT P10636 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PDE2A O00408 1/20 0.33
DPP4 P27487 1/20 0.32
DPP8 Q6V1X1 1/20 0.32
DPP9 Q86TI2 1/20 0.32
DPP7 Q9UHL4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL582147 0.99 SLC6A2 (0.35) SLC6A2SLC6A4SLC6A3CHRNA1CHRNG
Hydrochloric Acid SCHEMBL580625 0.86 SLC6A2 (0.37) SLC6A2SLC6A4SLC6A3CHRNA1CHRNG
SCHEMBL582145 0.85 SLC6A2 (0.37) SLC6A2SLC6A4SLC6A3CHRNA1CHRNG
SCHEMBL3063445 0.84 KDM1A (0.42) SLC6A2SLC6A4SLC6A3CHRNA1CHRNG
Hydrochloric Acid SCHEMBL581998 0.84 MAPT (0.32) MAPTTDP1
Hydrochloric Acid SCHEMBL580883 0.84 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3CHRNA1CHRNG
Hydrochloric Acid SCHEMBL580941 0.83 KDM1A (0.41) SLC6A2SLC6A4SLC6A3CHRNA1CHRNG
SCHEMBL581068 0.81 TDP1 (0.44) SLC6A2MAPTTDP1
Hydrochloric Acid SCHEMBL581553 0.81 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3CHRNA1CHRNG
SCHEMBL4505964 0.81 TDP1 (0.44) SLC6A2MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed