SCHEMBL5818031

SCHEMBL5818031

CON(C)C(=O)c1cc(C)n(Cc2ccccc2)n1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 10/20 0.47
CYP1A2 P05177 1/20 0.46
GAA P10253 2/20 0.45
RAB9A P51151 1/20 0.45
AURKA O14965 1/20 0.45
RPS6KB1 P23443 1/20 0.45
USP30 Q70CQ3 1/20 0.44
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
POLB P06746 1/20 0.43
P2RY14 Q15391 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21332671 0.88 HDAC3 (0.47) PTGER1GAARAB9AKMT2AMEN1
SCHEMBL4092138 0.83 PTGER1 (0.75) PTGER1
SCHEMBL22054628 0.81 GAA (0.59) PTGER1CYP1A2GAARAB9AAURKA
SCHEMBL6078431 0.81 AURKA (0.48) GAARAB9AAURKARPS6KB1KMT2A
SCHEMBL1137143 0.81 PTGER1 (0.59) PTGER1CYP1A2AURKARPS6KB1KMT2A
SCHEMBL5813326 0.81 SMYD3 (0.51) GAARAB9AKMT2AMEN1POLB
SCHEMBL9133656 0.80 PTGER1 (0.44) PTGER1CYP1A2AURKARPS6KB1USP30
SCHEMBL17324801 0.79 AURKA (0.52) PTGER1CYP1A2GAAAURKARPS6KB1
SCHEMBL1232379 0.78 PTGER1 (0.64) PTGER1CYP1A2GAAAURKARPS6KB1
SCHEMBL1233306 0.77 SMN1; SMN2 (0.60) PTGER1CYP1A2GAAAURKARPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006133885-A1 TRICYCLIC FUSED INDOLE DERIVATIVES AND THEIR USE AS AURORA KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2006-12-21 WO disclosed