SCHEMBL5819657

SCHEMBL5819657

Cc1nc(-c2nn(C3CCCCO3)cc2NC(=O)OC(C)(C)C)[nH]c1C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.37
HDAC4 P56524 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
ATR Q13535 3/20 0.32
FGFR1 P11362 1/20 0.32
DDR2 Q16832 1/20 0.32
BRAF P15056 1/20 0.32
RORC P51449 4/20 0.31
KDM5B Q9UGL1 1/20 0.31
KRAS P01116 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5578320 0.78 ABL1 (0.37) ABL1FGFR1DDR2BRAFRORC
SCHEMBL5812270 0.74 ABL1 (0.34) ABL1ATRFGFR1BRAFRORC
SCHEMBL5808054 0.74 ABL1 (0.34) ABL1HDAC4HDAC6ATRBRAF
SCHEMBL5821921 0.74 CNR2 (0.35) ABL1HDAC4HDAC6ATRBRAF
SCHEMBL5578291 0.74 ELANE (0.37) ABL1BRAF
SCHEMBL1645164 0.70 ATR (0.38) ABL1ATRBRAF
SCHEMBL2382993 0.70 ATR (0.36) ABL1ATRFGFR1DDR2BRAF
SCHEMBL14511713 0.69 CCNA2 (0.38) ABL1FGFR1DDR2BRAF
SCHEMBL30861007 0.69 BRD9 (0.37) ATRRORC
SCHEMBL4129018 0.68 NAMPT (0.36) ABL1ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006070202-A1 PYRAZOLE DERIVATIVES HAVING KINASE MODULATING ACTIVITY ASTEX THERAPEUTICS LIMITED (GB) 2006-07-06 WO disclosed