SCHEMBL5819952

SCHEMBL5819952

Cc1cnc(NC2CCC(NC(=O)c3ccc(F)c(F)c3)CC2)nc1NC1CC1

nearest known ligand 0.76

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 14/20 0.76
ADRA2A P08913 6/20 0.59
HRH1 P35367 6/20 0.59
HTR2B P41595 6/20 0.59
ADRA1A P35348 4/20 0.59
HTR1A P08908 1/20 0.55
NPY5R Q15761 1/20 0.55
KCNQ3 O43525 1/20 0.50
KCNQ2 O43526 1/20 0.50
AURKA O14965 2/20 0.49
AURKB Q96GD4 2/20 0.49
SYK P43405 1/20 0.48
MAPK14 Q16539 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6831616 0.94 MCHR1 (0.69) MCHR1ADRA2AHRH1HTR2BADRA1A
Trifluoroacetic Acid SCHEMBL6456478 0.94 MCHR1 (0.69) MCHR1ADRA2AHRH1HTR2BADRA1A
Trifluoroacetic Acid SCHEMBL6455569 0.89 MCHR1 (0.67) MCHR1ADRA2AHRH1HTR2BADRA1A
Trifluoroacetic Acid SCHEMBL6833473 0.89 MCHR1 (0.67) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL4258540 0.88 MCHR1 (0.71) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL4258534 0.88 MCHR1 (0.71) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6463341 0.87 MCHR1 (1.00) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6463334 0.87 MCHR1 (1.00) MCHR1ADRA2AHRH1HTR2BADRA1A
Trifluoroacetic Acid SCHEMBL6459409 0.86 MCHR1 (0.64) MCHR1ADRA2AHRH1HTR2BADRA1A
Trifluoroacetic Acid SCHEMBL6456496 0.86 MCHR1 (0.65) MCHR1ADRA2AHRH1HTR2BADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006091737-A1 MODULATORS OF GSK-3 ACTIVITY KEMIA, INC. (US) 2006-08-31 WO claimed