SCHEMBL5820378

SCHEMBL5820378

O=C(Cn1c2c(c3cc(Br)ccc31)CC(=O)Nc1ccccc1-2)NCCN1CCOCC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 8/20 0.64
CCNB2 O95067 7/20 0.62
CCNB1 P14635 7/20 0.62
GSK3B P49841 7/20 0.62
CCNB3 Q8WWL7 7/20 0.62
CNR2 P34972 3/20 0.45
KDM4E B2RXH2 3/20 0.43
RXFP1 Q9HBX9 1/20 0.43
HPGD P15428 2/20 0.43
GLA P06280 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KMT2A Q03164 3/20 0.43
POLB P06746 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MEN1 O00255 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
ABL1 P00519 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5819849 0.92 CDK1 (0.66) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5805246 0.85 CDK1 (0.73) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5802549 0.84 CDK1 (0.71) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5802581 0.82 CDK1 (0.69) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5801919 0.82 CDK1 (0.69) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5801923 0.80 CDK1 (0.79) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5819148 0.79 CDK1 (0.66) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5819011 0.79 CDK1 (0.55) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5688713 0.79 CDK1 (1.00) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5688439 0.77 GSK3B (1.00) CDK1CCNB2CCNB1GSK3BCCNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006089874-A1 BENZO[2,3]AZEPINO[4,5-B]INDOL-6-ONES GPC BIOTECH AG (DE) 2006-08-31 WO disclosed