SCHEMBL5821144

SCHEMBL5821144

COc1cccnc1C#Cc1csc(C)n1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 16/20 0.64
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4291588 0.78 GRM5 (1.00) GRM5
SCHEMBL4143647 0.78 GRM5 (1.00) GRM5CYP1A2CYP2D6
SCHEMBL4142443 0.75 GRM5 (1.00) GRM5CYP1A2CYP2D6
SCHEMBL15049682 0.74 GRM5 (1.00) GRM5CYP1A2CYP2D6
SCHEMBL4145767 0.73 GRM5 (0.72) GRM5CYP1A2CYP2D6
SCHEMBL1244096 0.72 GRM5 (0.67) GRM5CYP1A2CYP2D6
SCHEMBL1244088 0.72 GRM5 (0.66) GRM5
SCHEMBL5653763 0.71 GRM5 (0.70) GRM5CYP1A2CYP2D6
SCHEMBL14573619 0.71 GRM5 (0.70) GRM5CYP1A2CYP2D6
SCHEMBL4156970 0.71 GRM5 (1.00) GRM5CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1556142-A4 ALKYNE DERIVATIVES AS TRACERS FOR METABOTROPIC GLUTAMATE RECEPTOR BINDING MERCK & CO INC (US) 2006-11-08 EP disclosed
EP-1556142-A2 ALKYNE DERIVATIVES AS TRACERS FOR METABOTROPIC GLUTAMATE RECEPTOR BINDING Merck & Co., Inc. (US) 2005-07-27 EP disclosed
WO-2004038374-A2 ALKYNE DERIVATIVES AS TRACERS FOR METABOTROPIC GLUTAMATE RECEPTOR BINDING MERCK & CO., INC. (US) 2004-05-06 WO disclosed