SCHEMBL5823716

SCHEMBL5823716

COC(=O)c1cc(Oc2ccc(Nc3cc(-c4ccccc4)nc(Nc4ccccc4)n3)cc2)ccn1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BRAF P15056 7/20 0.49
SYK P43405 1/20 0.47
RAF1 P04049 3/20 0.44
P2RX3 P56373 5/20 0.44
MAPT P10636 1/20 0.44
IKBKB O14920 1/20 0.43
NFKB1 P19838 3/20 0.43
NR2C2 P49116 3/20 0.43
NFKB2 Q00653 3/20 0.43
RELA Q04206 3/20 0.43
TAB1 Q15750 3/20 0.43
JAK2 O60674 1/20 0.43
JAK3 P52333 1/20 0.43
VCP P55072 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1644392 0.89 AGPAT2 (0.51) BRAFRAF1P2RX3MAPT
SCHEMBL1644406 0.79 AGPAT2 (0.54) BRAFRAF1P2RX3MAPT
SCHEMBL3119465 0.78 AGPAT2 (0.53) BRAFRAF1P2RX3MAPTIKBKB
Hydrochloric Acid SCHEMBL3123797 0.78 AGPAT2 (0.53) BRAFRAF1P2RX3MAPT
SCHEMBL3119649 0.78 BRAF (0.58) BRAFRAF1NFKB1NR2C2NFKB2
SCHEMBL1643684 0.77 AGPAT2 (0.49) BRAFRAF1MAPT
SCHEMBL1642641 0.77 AGPAT2 (0.47) BRAFRAF1P2RX3MAPTIKBKB
SCHEMBL22737611 0.76 GCK (0.56) BRAFRAF1
SCHEMBL1644365 0.76 AGPAT2 (0.45) BRAFRAF1MAPT
SCHEMBL1643674 0.75 MCL1 (0.47) BRAFP2RX3MAPTIKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689722-A2 4-AMINOPYRIMIDINE DERIVATIVES FOR TREATMENT OF HYPERPROLIFERATIVE DISORDERS Bayer Pharmaceuticals Corporation (US) 2006-08-16 EP disclosed
WO-2005035507-A2 4-AMINOPYRIMIDINE DERIVATIVES FOR TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER PHARMACEUTICALS CORPORATION (US) 2005-04-21 WO disclosed