SCHEMBL5825867

SCHEMBL5825867

COc1cc2nccc(Oc3ccccc3S(=O)(=O)CCOc3ccc(C)cc3)c2cc1OC

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 2/20 0.51
KDR P35968 1/20 0.51
AXL P30530 4/20 0.50
SRC P12931 4/20 0.49
TGFBR1 P36897 4/20 0.49
PDGFRB P09619 1/20 0.48
FGFR2 P21802 2/20 0.47
MET P08581 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5825071 0.85 PDGFRA (0.59) PDGFRAKDRSRCTGFBR1PDGFRB
SCHEMBL5824451 0.79 PDGFRA (0.66) PDGFRAKDRPDGFRBFGFR2
SCHEMBL5825445 0.78 PDGFRA (0.59) PDGFRAKDRAXLSRCPDGFRB
SCHEMBL5824390 0.76 AXL (0.56) PDGFRAKDRAXLPDGFRBFGFR2
SCHEMBL12444104 0.76 PDGFRA (0.76) PDGFRAKDRPDGFRBFGFR2
SCHEMBL5826205 0.75 PDGFRA (0.52) PDGFRAKDRAXLSRCTGFBR1
SCHEMBL5824511 0.75 PDGFRA (0.56) PDGFRAKDRPDGFRBFGFR2
SCHEMBL5825827 0.74 FGFR2 (0.63) PDGFRAKDRAXLPDGFRBFGFR2
SCHEMBL5825801 0.74 PDGFRA (0.66) PDGFRAKDRPDGFRBFGFR2
SCHEMBL5824659 0.74 FGFR2 (0.50) PDGFRAKDRAXLPDGFRBFGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7135466-B2 Quinoline and quinazoline derivatives and drugs containing the same KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-14 US claimed